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Nov 08, 2022

Qee qhov kev qhia txog lappaconitine hydrobromide

Lappaconitine hydrobromide

Bioactivity

Kev piav qhia

Lappaconitine hydrobromideyogib tug natural alkaloid compound nrog antiarrhythmic zog.

Solubility

In vitro: 10mM hauv DMSOLappaconitine Hydrobromide

Tshuag daws

1 mM 1.5024 mL 7.5119 mL 15.0238 mL

5 mM 0.3005 mL 1.5024 mL 3.0048 mL

1 0 mM 0.1502 mL 0.7512 mL 1.5024 mL

Chemical thiab Physical Properties

Boiling point

740.8ºC ntawm 760 mmHg

Melting point

223-226ºC

Cov mis mos molecular

C32H45BrN2O8

Molecular hnyav

665.612

Flash point

401.8ºC

Cov huab hwm coj

664.235901

PSA

126.79000

LogP

3.19060

Qhov tshwm sim

hmoov dawb

Cia tej yam kev mob

2-8 degree




Pharmacological kev ua

Lappaconitine hydrobromide yog ib qho tshuaj analgesic uas tsis muaj tshuaj lom nrog cov nyhuv analgesic. Cov khoom no kuj muaj tshuaj loog hauv zos, ua kom txias, antipyretic thiab anti-inflammatory teebmeem. Piv nrog pethidine, cov nyhuv analgesic ntawm cov khoom no yog sib npaug, lub sij hawm pib qeeb me ntsis, thiab lub sij hawm txij nkawm ntev dua; cov nyhuv analgesic yog 7 npaug ntawm cov tshuaj antipyretic analgesic aminopyrine.






Specification
90-99 feem pua




Peb qhov zoo
1.Kev xa khoom sai.Kev lees paub zoo2.Our R & D pab neeg yog tsim los ntawm post-doctoral, biological thiab zaub mov kawm tiav nrog ywj siab, R & D muaj peev xwm.3. Muab cov kev pabcuam ntim khoom customized.OEM kev pabcuam suav nrog: softgel, capsule, ntsiav tshuaj, hnab, granule, thiab lwm yam. Kev pabcuam rautsim cov neeg siv khoom tshwj xeeb nrog ntau tshaj 100 tus neeg siv khoom thoob ntiaj teb.4.Over 10 xyoo dhau los hauv herballngrents ntau lawm raws li GMPstandard. Tag nrho cov kev paub ntawm tshuaj ntsuab extracts zoo tswj thiab daim ntawv thov.




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