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Apr 20, 2023

Cov teebmeem pharmacological thiab cov piv txwv soj ntsuam ntawm Lappaconitine Hydrobromide

 

Lappaconitine Hydrobromide(Cov ntawv luv:LH) yog ib yam tshuaj uas siv tau los kho ntau yam kab mob. Nws belongs rau acrylic NSAIDs thiab feem ntau yog siv los txo qhov mob me mus rau nruab nrab, xws li mob taub hau, mob hniav, thiab mob cov tsos mob xws li mob caj dab.

Ntxiv rau,LHmuaj lwm yam teebmeem tshuaj, xws li tshuaj tiv thaiv kab mob, tshuaj tiv thaiv platelet, antipyretic, thiab lwm yam, yog li nws tau siv dav hauv kev kho mob sib txawv hauv kev kho mob.

Hauv qab no yog cov teebmeem pharmacological thiab cov piv txwv ntawm kev kho mobLH:

 

Lappaconitine Hydrobromide

 

 

Cov nyhuv analgesic

 

 

LHexerts analgesic nyhuv tsuas yog los ntawm inhibiting cyclooxygenase (COX). COX yog ib qho enzyme uas hloov ferulic acid rau hauv prostaglandins thiab lwm yam tshuaj. Thaum cov ntaub so ntswg ntawm lub cev khaus, COX tso tawm cov tshuaj uas ua rau cov hlab ntsha tawg thiab ua rau muaj mob hauv zos uas tuaj yeem ua rau mob.

Yog li ntawd, inhibiting cov haujlwm ntawm COX tuaj yeem txo qis qhov mob thiab yog li txo qhov mob.

Clinical piv txwv:LHtuaj yeem siv los txo cov tsos mob xws li mob taub hau, mob hniav, mob khaub thuas, mob nqaij, thiab mob caj dab.

 

 

Anti-inflammatory nyhuv

 

 

LHmuaj peev xwm inhibit zus tau tej cov tshuaj nyob rau hauv inflammatory hlwb, txo o, thiab txo cov tsos mob xws li liab, o thiab mob. Cov tshuaj no tuaj yeem tiv thaiv kev hloov pauv ntawm lub zog ntawm NF-κB thiab tiv thaiv nws cov nyhuv anti-inflammatory.

Clinical piv txwv:LHtuaj yeem siv los kho cov kab mob xws li mob caj dab rheumatoid, ankylosing spondylitis, thiab cervical spondylitis.

 

 

Cov nyhuv antiplatelet

 

 

LHtuaj yeem tiv thaiv platelet aggregation, yog li txo qhov muaj peev xwm ntawm thrombosis. Cov tshuaj no ua rau nws cov nyhuv antiplatelet los ntawm inhibiting cov synthesis ntawm thromboxane thiab arachidonic acid.

Clinical piv txwv:LHtuaj yeem siv los tiv thaiv cov kab mob thrombotic xws li myocardial infarction thiab mob stroke.

 

 

Antipyretic nyhuv

 

 

LHtuaj yeem ua kom cov nyhuv antipyretic los ntawm inhibiting zus tau tej cov prostaglandins. Prostaglandins yog cov tshuaj uas tuaj yeem ua rau koj lub cev kub thiab ua rau kub taub hau.

Clinical piv txwv:LHsiv tau los kho kub taub hau, xws li mob khaub thuas, mob khaub thuas thiab lwm yam tsos mob.

 

 

Anti-tumor nyhuv

 

 

LHtuaj yeem siv los tiv thaiv qog nqaij hlav los ntawm cov txheej txheem sib txawv. Piv txwv li, nws muaj peev xwm inhibit qog cell proliferation thiab metastasis, thiab txhawb cov qog cell apoptosis.

Clinical piv txwv:LHyog siv los kho qee cov qog nqaij hlav, xws li mob cancer mis thiab mob plab.

 

 

Immunomodulatory

 

 

LHtuaj yeem txo cov lus teb inflammatory thiab txhim khu kev ua haujlwm ntawm lub cev tiv thaiv kab mob los ntawm inhibiting lub zais ntawm cov hlwb inflammatory.

Clinical piv txwv:LHtuaj yeem siv los kho cov kab mob tiv thaiv kab mob xws li mob rheumatism thiab kab mob lupus erythematosus.

 

Feem ntau,LHmuaj ntau yam teebmeem pharmacological thiab siv dav hauv kev kho mob ntawm cov tsos mob sib txawv thiab kab mob. Txawm li cas los xij, siv nws nrog ceev faj thiab ua raws li koj tus kws kho mob cov lus qhia thiab ntau npaum li cas kom tsis txhob muaj qhov tshwm sim tsis zoo.

 

 

Khoom Description

 

 

KINTA yog lub chaw tsim khoom tshwj xeeb hauv kev tsim cov khoom siv tshuaj lom neeg, uas nws cov khoom tau siv dav hauv kev lag luam tshuaj thiab lwm yam lag luam. Lub purity ntawm LH tsim los ntawm KINTA yog siab li 99 feem pua. Nws yog cov khoom siv tshuaj nquag siv, thiab nws txoj kev siv tseem ceeb yog cov tshuaj nruab nrab.

 

Nrog rau qhov zoo, kev sib tw nqi thiab kev pabcuam, peb cov khoom tau yeej lub koob npe nrov thiab lub koob npe nrov hauv kev lag luam txawv teb chaws. KINTAI ua raws li kev coj noj coj ua ntawm cov neeg ua haujlwm zoo thiab tau cog lus los txhim kho cov khoom zoo thiab txo cov nqi. Nrog rau txoj kev loj hlob yav tom ntej, KINTAI yuav txuas ntxiv mus nrhiav kev lag luam lub tswv yim ntawm "zoo li cov tub ntxhais thiab cov neeg siv khoom ua qhov chaw", txuas ntxiv tsim kho tshiab thiab ua kom zoo dua qub, thiab muab cov neeg siv khoom zoo dua thiab cov kev pabcuam zoo dua.

 

Yog tias koj xav paub ntau ntxiv txog Lappaconitine Hydrobromide, thov koj xav tiv tauj peb ntawmsales@kintaibio.comlos yog tawm tswv yim nyob rau nplooj ntawv tom ntej.

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